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Moynihan & Crean: The Physicochemical Basis of Pharmaceuticals

Hyperlinked bibliography

Click on the links below to view the references from the book with active links to online journal articles, where available. Please note that some of the sites you will be directed to may require a username and password to access the full text article.

Chapter 1

FDA (Food and Drug Administration). (2004). Innovation or stagnation: Challenge and opportunity on the critical path to new medical products. [http://www.fda.gov/ScienceResearch/SpecialTopics/CriticalPathInitiative/CriticalPathOpportunitiesReports/ucm077262.htm]

Lipinski, C. A. et al. (2001). Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings. Advanced Drug Delivery Review, 46, 3–26. [DOI: 10.1016/S0169-409X(00)00129-0] [PubMed: 11259830]

Chapter 2

Bell, R. P. (1973) The Proton in Chemistry (2nd edn) London: Chapman and Hall.

Eisenberg, D., and Kauzmann, W. (1969). The Structure and Properties of Water. Oxford University Press.

Frank, H. S. (1970). Science, 169, 635. [DOI: 10.1126/science.169.3946.635] [PubMed: 17791838]

Garrett, E. R. (1957). J. Am. Chem. Soc., 79, 3401. [DOI: 10.1021/ja01570a024]

Chapter 3

Abraham, H. A. et al. (2008). Eur. J. Med. Chem. 43, 478–485. [DOI: 10.1016/j.ejmech.2007.04.002] [PubMed: 17544548]

Alberty, R. A., and Silbey, R. J. (1992). Physical Chemistry. New York: John Wiley & Sons.

Burger, A. (1982). Acta Pharm. Tech., Vol. 28(1), 1–20.

Chickos, J. S., and Acree, W. E. (2003). J. Phys. Chem. Ref. Data, Vol. 32(2), 519–879. [DOI: 10.1063/1.1529214]

Chapter 4

Bingham, A. L., Hughes, D. S., Hursthouse, M. B., Lancaster, R. W., Tavener, S., Threlfall, T. L. (2001) Over one hundred solvates of sulfathiazole. Chem. Commun., 603–604. [DOI: 10.1039/b009540k]

Blagden, N. (2001) Crystal engineering of polymorph appearance: the case of sulfathiazole. Powder Technology, 121, 46–52. [DOI: 10.1016/S0032-5910(01)00373-4]

British Pharmacopoeia (2008), The Stationery Office, London.

Chemburkar S. R., Bauer J., Deming K., Spiwek H., Patel K., Morris J., Henry R., Spanton S., Dziki W., Porter W., Quick J., Bauer P., Donaubauer J., Narayanan B. A., Soldani M., Riley D., McFarland K. (2000) Dealing with the Impact of Ritonavir Polymorphs on the Late Stages of Bulk Drug Process Development. Organic Process Research and Development, 4, 413–417. [DOI: 10.1021/op000023y]

Joiris, E., Di Martino, P., Berneron, C., Guyot-Hermann, A.-M., Guyot, J.-C. (1998) The compression behaviour of orthorhombic paracetamol. Pharm. Res., 15, 1122–1130. [DOI: 10.1023/A:1011954800246] [PubMed: 9688070]

Leadbeater, C. (1991) Glaxo fights for zantac patent, Financial Times, Tuesday, April 9.

Chapter 5

Barnes, G.T. and Gentle, I.R. (2005). Interfacial Science. Oxford University Press, Oxford.

Griffin, W.C. (1949). Classification of surface-active agents by HLB, Journal of the Society of Cosmetic Chemists 1, 311–326.

Chapter 7

Demare, S., Slater, B., Lacombe, G., Breuzin, D., Dini, C. (2007) Accurate automated log Po/w measurement by gradient-flow liquid-liquid partition chromatography, J. Chromatography A, 1175, 16–25. [DOI: 10.1016/j.chroma.2007.09.093]

Frum, Y., Khan, G. M., Sefcik, J., Rouse, J., Eccleston, G. M. and Meidan, V. M.(2007), Towards a correlation between drug properties and in vitro transdermal flux variability. Int. J. Pharm., 336, 140–147 [DOI: 10.1016/j.ijpharm.2006.11.049] [PubMed: 17182201]

Leo, A. L. (1990) Method of Calculating Partition Coefficients, from Comprehensive Medicinal Chemistry, Vol. 4, C. Hansch, P. G. G. Sammes and J. B. Taylor (eds), C. A. Ramsden (Vol. Ed.), pp 295–319

Michalets, E. L. (1998) Update: Clinically significant cytochrome P-450 drug interactions, Pharmacotherapy, 18, 86–112

Mirrlees, M. S., Moulton, S. J., Murphy, C. T., Taylor, P. J. (1976) Direct Measurement of Octanol-Water Partition Coefficients by High-Pressure Liquid Chromatography, J. Med. Chem., 19, 615–619 [DOI: 10.1021/jm00227a008] [PubMed: 1271403]